Monday, February 24, 2014

Witting Reaction

The Witting Reaction:

  •  Witting reaction is an important method of preparation of alkene from aldehyde or ketone.
  • This reaction was discovered by the scientist Georg Witting in 1954, for which he was awarded the Nobel Prize in Chemistry in 1979.

In this reaction, when an aldehyde or ketone reacts with a triphenyl phosphonium ylide, it gives out substituted alkene and triphenyl phosphine oxide.



Example of witting reaction:
There are few examples of witting reaction.




Mechanism of witting reaction:

Witting reaction is carried out under mild condition. It is basically a three steps process.

Step I: In step I when a carbonyl compound reacts with ylide, a dipolar charge-seperated species betaine is formed.



Step II: With rearrangement, betaine is converted into four membered heterocyclic structure which is called as an oxaphosphatane.



Step III: Cleaveage of oxaphosphatane takes place which leads to alkene and phosphine oxide as products.



What is ylide?

Triphenyl phosphonium ylide is also known as witting reagent. It is a neutral molecule but have positive and negative centres on the adjacent atoms that are connected by a sigma ( ) bond.  

The ylides is prepared in two steps:

1. SN2 reaction between triphenyl phosphine and an alkyl halide
2. Abstraction of a proton by a strong base



The mechanism of the reaction is given follow:

1.



2.

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